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Kazuaki Niikura Selected Research

2,6- dichloro- N- (1- (2- (4- morpholinyl)- 2- oxoethyl)- 2- (trifluoromethyl)- 1H- benzimidazol- 4- yl)benzamide

4/2007FR177995, a novel vacuolar ATPase inhibitor, exerts not only an inhibitory effect on bone destruction but also anti-immunoinflammatory effects in adjuvant-induced arthritic rats.

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Kazuaki Niikura Research Topics

Disease

7Bone Resorption
09/2007 - 06/2004
3Bone Diseases (Bone Disease)
04/2007 - 06/2004
2Hypercalcemia (Milk Alkali Syndrome)
04/2007 - 09/2005
1Pain (Aches)
01/2017
1Breast Neoplasms (Breast Cancer)
09/2007
1Osteolysis
09/2007
1Neoplasm Metastasis (Metastasis)
09/2007
1Neoplasms (Cancer)
09/2007
1Arthritis (Polyarthritis)
04/2007
1Rheumatoid Arthritis
04/2007
1Inflammation (Inflammations)
04/2007
1Osteopetrosis
04/2006
1Periodontal Diseases (Periodontal Disease)
12/2005
1Periodontitis
12/2005
1Alveolar Bone Loss
12/2005
1Body Weight (Weight, Body)
09/2005

Drug/Important Bio-Agent (IBA)

6Adenosine Triphosphatases (ATPase)IBA
09/2007 - 06/2004
4Vacuolar Proton-Translocating ATPases (V-Type ATPase)IBA
09/2007 - 06/2004
22,6- dichloro- N- (3- methyl- 4- (3- methyl- 2- oxo- 1- imidazolidinyl)- 8- quinolinyl)benzamideIBA
09/2007 - 12/2005
2Interleukin-1 (Interleukin 1)IBA
04/2007 - 09/2005
2Pharmaceutical PreparationsIBA
04/2007 - 06/2004
2Interleukin-6 (Interleukin 6)IBA
04/2007 - 09/2005
2Tretinoin (Retinoic Acid)FDA LinkGeneric
04/2007 - 09/2005
2FR 167356IBA
09/2005 - 06/2004
1salicylhydroxamic acid (SHAM)IBA
01/2017
1GlycosaminoglycansIBA
04/2007
12,6- dichloro- N- (1- (2- (4- morpholinyl)- 2- oxoethyl)- 2- (trifluoromethyl)- 1H- benzimidazol- 4- yl)benzamideIBA
04/2007
1N-Acetylneuraminic Acid (Sialic Acid)IBA
04/2007
1Diphosphonates (Bisphosphonates)IBA
02/2007
1apicularen AIBA
02/2007
1cimadronateIBA
02/2007
1Dihydrotachysterol (AT 10)IBA
02/2007
1Interleukin-1beta (Interleukin 1 beta)IBA
02/2007
1apicularen BIBA
02/2007
1Parathyroid Hormone (Parathormone)IBA
02/2007
1oxidized low density lipoproteinIBA
06/2004

Therapy/Procedure

1Oral Administration
12/2005
1Ligation
12/2005